Page 19 - Read Online

Ji et al. Chem Synth 2022;2:17 https://dx.doi.org/10.20517/cs.2022.27 Page 11 of 11

drug design and discovery. J Med Chem 2014;57:2832-42. DOI PubMed
19. Feng M, Tang B, Liang SH, Jiang X. Sulfur containing scaffolds in drugs: synthesis and application in medicinal chemistry. Curr Top
Med Chem 2016;16:1200-16. DOI PubMed PMC
20. Scott KA, Njardarson JT. Analysis of US FDA-approved drugs containing sulfur atoms. Top Curr Chem (Cham) 2018;376:5. DOI
PubMed
21. Giannetti AM, Wong H, Dijkgraaf GJ, et al. Identification, characterization, and implications of species-dependent plasma protein
binding for the oral Hedgehog pathway inhibitor vismodegib (GDC-0449). J Med Chem 2011;54:2592-601. DOI PubMed
22. Tsui GC, Lautens M. Linear-selective rhodium(I)-catalyzed addition of arylboronic acids to allyl sulfones. Angew Chem Int Ed Engl
2010;49:8938-41. DOI PubMed
23. Nishimura T, Takiguchi Y, Hayashi T. Effect of chiral diene ligands in rhodium-catalyzed asymmetric addition of arylboronic acids to
α,β-unsaturated sulfonyl compounds. J Am Chem Soc 2012;134:9086-9. DOI PubMed
24. So CM, Kume S, Hayashi T. Rhodium-catalyzed asymmetric hydroarylation of 3-pyrrolines giving 3-arylpyrrolidines: protonation as a
key step. J Am Chem Soc 2013;135:10990-3. DOI PubMed
25. Lim KM, Hayashi T. Rhodium-catalyzed asymmetric arylation of allyl sulfones under the conditions of isomerization into alkenyl
sulfones. J Am Chem Soc 2015;137:3201-4. DOI PubMed
26. Yan Q, Xiao G, Wang Y, Zi G, Zhang Z, Hou G. Highly efficient enantioselective synthesis of chiral sulfones by Rh-catalyzed
asymmetric hydrogenation. J Am Chem Soc 2019;141:1749-56. DOI PubMed
27. Oxtoby LJ, Gurak JA Jr, Wisniewski SR, Eastgate MD, Engle KM. Palladium-catalyzed reductive heck coupling of alkenes. Trends
Chem 2019;1:572-87. DOI PubMed PMC
28. Tao ZL, Adili A, Shen HC, Han ZY, Gong LZ. Catalytic enantioselective assembly of homoallylic alcohols from dienes,
aryldiazonium salts, and aldehydes. Angew Chem Int Ed Engl 2016;55:4322-6. DOI PubMed
29. Zhang T, Li WA, Shen HC, Chen SS, Han ZY. Chiral-anion-mediated asymmetric heck-matsuda reaction of acyclic alkenyl alcohols.
Org Lett 2021;23:1473-7. DOI PubMed
30. Werner EW, Sigman MS. Operationally simple and highly (E)-styrenyl-selective Heck reactions of electronically nonbiased olefins. J
Am Chem Soc 2011;133:9692-5. DOI PubMed PMC
31. Zong Y, Hu J, Sun P, Jiang X. Synthesis of biaryl derivatives via a magnetic Pd-NPs-catalyzed one-pot diazotization - cross-coupling
reaction. Synlett 2012;23:2393-6. DOI
32. CCDC 2152365 (5p) contains the supplementary crystallographic data for this paper. More detail, see supporting information chapter
6. The data can be obtained free of charge from The Cambridge Crystallographic Data Centre. Available from:
www.ccdc.cam.ac.uk/structures [Last accessed on 12 Oct 2022].
33. Lin Y, Kuo Y, Kuei C, Chang M. Palladium-mediated synthesis of 1,1,2-triarylethanes. Application to the synthesis of CDP-840.
Tetrahedron 2017;73:1275-82. DOI
34. Liang Q, Walsh PJ, Jia T. Copper-catalyzed intermolecular difunctionalization of styrenes with thiosulfonates and arylboronic acids
via a radical relay pathway. ACS Catal 2020;10:2633-9. DOI