Page 26 - Read Online
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Page 22 of 23          Skoreński et al. Rare Dis Orphan Drugs J 2023;2:6  https://dx.doi.org/10.20517/rdodj.2022.21

                   64.  DOI  PubMed
               33.      Wysocka M, Lesner A, Gruba N, et al. Three wavelength substrate system of neutrophil serine proteinases. Anal Chem 2012;84:7241-
                   8.  DOI  PubMed
               34.      Sun Q, Li J, Liu WN, Dong QJ, Yang WC, Yang GF. Non-peptide-based fluorogenic small-molecule probe for elastase. Anal Chem
                   2013;85:11304-11.  DOI  PubMed
               35.      Aikawa N, Kawasaki Y. Clinical utility of the neutrophil elastase inhibitor sivelestat for the treatment of acute respiratory distress
                   syndrome. Ther Clin Risk Manag 2014;10:621-9.  DOI  PubMed  PMC
               36.      Powers JC, Gupton BF, Harley AD, Nishino N, Whitley RJ. Specificity of porcine pancreatic elastase, human leukocyte elastase and
                   cathepsin G. Inhibition with peptide chloromethyl ketones. Biochim Biophys Acta 1977;485:156-66.  DOI  PubMed
               37.      Jugniot N, Voisin P, Bentaher A, Mellet P. Neutrophil elastase activity imaging: recent approaches in the design and applications of
                   activity-based probes and substrate-based probes. Contrast Media Mol Imaging 2019;2019:7417192.  DOI  PubMed  PMC
               38.      Winiarski Ł, Oleksyszyn J, Sieńczyk M. Human neutrophil elastase phosphonic inhibitors with improved potency of action. J Med
                   Chem 2012;55:6541-53.  DOI  PubMed
               39.      António JPM, Gonçalves LM, Guedes RC, Moreira R, Gois PMP. Diazaborines as new inhibitors of human neutrophil elastase. ACS
                   Omega 2018;3:7418-23.  DOI  PubMed  PMC
               40.      Zheng Q, Woehl JL, Kitamura S, et al. SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase. Proc
                   Natl Acad Sci USA 2019;116:18808-14.  DOI  PubMed  PMC
               41.      Xu Y, Qi N, Wen H, Zhang G, Wang Y, Cui H. Synthesis and evaluation of benzenesulfonic acid derivatives as human neutrophil
                   elastase (hNE) inhibitors. Med Chem Res 2021;30:387-98.  DOI  PubMed  PMC
               42.      Al-Horani RA, Aliter KF, Kar S, Mottamal M. Sulfonated nonsaccharide heparin mimetics are potent and noncompetitive inhibitors of
                   human neutrophil elastase. ACS Omega 2021;6:12699-710.  DOI  PubMed  PMC
               43.      Ruivo EF, Gonçalves LM, Carvalho LA, et al. Clickable 4-Oxo-β-lactam-based selective probing for human neutrophil elastase related
                   proteomes. ChemMedChem 2016;11:2037-42.  DOI  PubMed
               44.      Schulz-Fincke AC, Tikhomirov AS, Braune A, et al. Design of an activity-based probe for human neutrophil elastase: implementation
                   of the lossen rearrangement to induce förster resonance energy transfers. Biochemistry 2018;57:742-52.  DOI  PubMed
               45.      Anderson BM, Poole DP, Aurelio L, et al. Application of a chemical probe to detect neutrophil elastase activation during inflammatory
                   bowel disease. Sci Rep 2019;9:13295.  DOI  PubMed  PMC
               46.      Liu SY, Xiong H, Li RR, Yang WC, Yang GF. Activity-based near-infrared fluorogenic probe for enabling in vitro and in vivo
                   profiling of neutrophil elastase. Anal Chem 2019;91:3877-84.  DOI  PubMed
               47.      Ahmad S, Saleem M, Riaz N, et al. The natural polypeptides as significant elastase inhibitors. Front Pharmacol 2020;11:688.  DOI
                   PubMed  PMC
               48.      Marinaccio L, Stefanucci A, Scioli G, et al. Peptide human neutrophil elastase inhibitors from natural sources: an overview. Int J Mol
                   Sci 2022;23:2924.  DOI  PubMed  PMC
               49.      Wan H, Lee KS, Kim BY, et al. A spider-derived Kunitz-type serine protease inhibitor that acts as a plasmin inhibitor and an elastase
                   inhibitor. PLoS One 2013;8:e53343.  DOI  PubMed  PMC
               50.      Luan N, Zhao Q, Duan Z, et al. Identification and characterization of ShSPI, a Kazal-type elastase inhibitor from the venom of
                   scolopendra hainanum. Toxins (Basel) 2019;11:708.  DOI  PubMed  PMC
               51.      Al-Awadhi FH, Paul VJ, Luesch H. Structural diversity and anticancer activity of marine-derived elastase inhibitors: key features and
                   mechanisms mediating the antimetastatic effects in invasive breast cancer. Chembiochem 2018;19:815-25.  DOI  PubMed  PMC
               52.      Luo D, Luesch H. Ahp-cyclodepsipeptide inhibitors of elastase: lyngbyastatin 7 stability, scalable synthesis, and focused library
                   analysis. ACS Med Chem Lett 2020;11:419-25.  DOI  PubMed  PMC
               53.      Keller L, Canuto KM, Liu C, et al. Tutuilamides A-C: vinyl-chloride-containing cyclodepsipeptides from marine cyanobacteria with
                   potent elastase inhibitory properties. ACS Chem Biol 2020;15:751-7.  DOI  PubMed  PMC
               54.      Crisford H, Sapey E, Stockley RA. Proteinase 3; a potential target in chronic obstructive pulmonary disease and other chronic
                   inflammatory diseases. Respir Res 2018;19:180.  DOI  PubMed  PMC
               55.      Korkmaz B, Lesner A, Guarino C, et al. Inhibitors and antibody fragments as potential anti-inflammatory therapeutics targeting
                   neutrophil proteinase 3 in human disease. Pharmacol Rev 2016;68:603-30.  DOI  PubMed
               56.      Grzywa R, Lesner A, Korkmaz B, Sieńczyk M. Proteinase 3 phosphonic inhibitors. Biochimie 2019;166:142-9.  DOI  PubMed
               57.      Witko-Sarsat V, Thieblemont N. Granulomatosis with polyangiitis (Wegener granulomatosis): a proteinase-3 driven disease? Joint
                   Bone Spine 2018;85:185-9.  DOI  PubMed
               58.      Epinette C, Croix C, Jaquillard L, et al. A selective reversible azapeptide inhibitor of human neutrophil proteinase 3 derived from a
                   high affinity FRET substrate. Biochem Pharmacol 2012;83:788-96.  DOI  PubMed
               59.      Popow-Stellmaszyk J, Wysocka M, Lesner A, Korkmaz B, Rolka K. A new proteinase 3 substrate with improved selectivity over
                   human neutrophil elastase. Anal Biochem 2013;442:75-82.  DOI  PubMed
               60.      Guarino C, Legowska M, Epinette C, et al. New selective peptidyl di(chlorophenyl) phosphonate esters for visualizing and blocking
                   neutrophil proteinase 3 in human diseases. J Biol Chem 2014;289:31777-91.  DOI  PubMed  PMC
               61.      Guarino C, Gruba N, Grzywa R, et al. Exploiting the S4-S5 specificity of human neutrophil proteinase 3 to improve the potency of
                   peptidyl di(chlorophenyl)-phosphonate ester inhibitors: a kinetic and molecular modeling analysis. J Med Chem 2018;61:1858-70.
                   DOI  PubMed
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